1,3,5-Trimethoxy-2-(2-nitrovinyl)benzene [C11H13NO5]

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Results

Date

2 substances in Reaxys

2018-07-09 14h:39m:23s (UTC)

O

1. Query

O

O N

O

O

Search as: As drawn ))

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2018-07-09 14:42:02


Reaxys ID 3145953 View in Reaxys

O

1/2 Chemical Name: (E)-1,3,5-trimethoxy-2-(2-nitrovinyl)benzene; (E)-2,4,6-trimethoxy-β-nitrostyrene; 2,4,6-trimethoxy-β-nitrostyrene; (E)-2,4,6-trimethoxy-β-nitro-styrene; (E)-2,4,6-Trimethoxy-β-nitro-styrol Linear Structure Formula: C11H13NO5 Molecular Formula: C11H13NO5 Molecular Weight: 239.228 Type of Substance: isocyclic InChI Key: URHPFHDNYKOMAI-SNAWJCMRSA-N Note:

O N

O

O

O

Substance Label (4) Label References 3b

Zhang, Min; Hu, Peng; Zhou, Jun; Wu, Ge; Huang, Shijun; Su, Weiping; Organic Letters; vol. 15; nb. 7; (2013); p. 1718 - 1721, View in Reaxys

5b

Suzuki, Tomiko M.; Yamamoto, Masami; Fukumoto, Keiko; Akimoto, Yusuke; Yano, Kazuhisa; Journal of Catalysis; vol. 251; nb. 2; (2007); p. 249 - 257, View in Reaxys

6d

Fedou, Nicolas M.; Parsons, Philip J.; Viseux, Eddy M. E.; Whittle, Alan J.; Organic Letters; vol. 7; nb. 15; (2005); p. 3179 - 3182, View in Reaxys

3h

Liu, Ju-Tsung; Yao, Ching-Fa; Tetrahedron Letters; vol. 42; nb. 35; (2001); p. 6147 - 6150, View in Reaxys

Druglikeness (1) 1 of 1

LogP

2.242

H Bond Donors

0

H Bond Acceptors

0

Rotatable Bonds

5

TPSA

73.51

Lipinski Number

4

Veber Number

2

Melting Point (1) 1 of 1

Melting Point [°C]

177 - 177.5

Solvent (Melting Point)

ethanol

Benington et al.; Journal of Organic Chemistry; vol. 19; (1954); p. 11,14, View in Reaxys Crystal Property Description (3) Colour & Other Location Properties

References

yellow

supporting informa- Zhang, Min; Hu, Peng; Zhou, Jun; Wu, Ge; Huang, Shijun; Su, Weiping; Organic Letters; tion vol. 15; nb. 7; (2013); p. 1718 - 1721, View in Reaxys

yellow

supporting informa- Zhang, Min; Zhou, Jun; Kan, Jian; Wang, Min; Su, Weiping; Hong, Maochun; Chemical tion Communications; vol. 46; nb. 30; (2010); p. 5455 - 5457, View in Reaxys

gelb

Benington et al.; Journal of Organic Chemistry; vol. 19; (1954); p. 11,14, View in Reaxys

NMR Spectroscopy (3) 1 of 3

Description (NMR Spectroscopy)

Chemical shifts; Spectrum

Nucleus (NMR Spectroscopy)

1H

Solvents (NMR Spectroscopy)

chloroform-d1

Frequency (NMR Spectro- 400 scopy) [MHz] Location

supporting information

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2/10

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Zhang, Min; Zhou, Jun; Kan, Jian; Wang, Min; Su, Weiping; Hong, Maochun; Chemical Communications; vol. 46; nb. 30; (2010); p. 5455 - 5457, View in Reaxys; Zhang, Min; Hu, Peng; Zhou, Jun; Wu, Ge; Huang, Shijun; Su, Weiping; Organic Letters; vol. 15; nb. 7; (2013); p. 1718 - 1721, View in Reaxys 2 of 3

Description (NMR Spectroscopy)

Chemical shifts; Spectrum

Nucleus (NMR Spectroscopy)

13C

Solvents (NMR Spectroscopy)

chloroform-d1

Frequency (NMR Spectro- 101 scopy) [MHz] Location

supporting information

Zhang, Min; Hu, Peng; Zhou, Jun; Wu, Ge; Huang, Shijun; Su, Weiping; Organic Letters; vol. 15; nb. 7; (2013); p. 1718 1721, View in Reaxys 3 of 3

Description (NMR Spectroscopy)

Chemical shifts; Spectrum

Nucleus (NMR Spectroscopy)

13C

Solvents (NMR Spectroscopy)

chloroform-d1

Frequency (NMR Spectro- 100 scopy) [MHz] Location

supporting information

Zhang, Min; Zhou, Jun; Kan, Jian; Wang, Min; Su, Weiping; Hong, Maochun; Chemical Communications; vol. 46; nb. 30; (2010); p. 5455 - 5457, View in Reaxys Medchem (21) 1 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Minimum inhibitory concentration of the compound dissolved in DMSO against Stenotrophomonas maltophilia ATCC 13637 by disk diffusion susceptibility assay

Biological Species/NCBI ID

Stenotrophomonas maltophilia ATCC 13637

Substance RN

3145953View in Reaxys

Measurement Parameter

MIC

Unit

µg

Measurement Object

Minimum Inhibitory Concentration

Qualitative value

>

Quantitative value

100

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 2 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Minimum inhibitory concentration of the compound dissolved in DMSO against Escherichia coli ATCC 25922 by disk diffusion susceptibility assay

Biological Species/NCBI ID

Escherichia coli ATCC 25922

Substance RN

3145953View in Reaxys

Measurement Parameter

MIC

Unit

µg

Measurement Object

Minimum Inhibitory Concentration

Qualitative value

>

Copyright © 2018 Elsevier Life Sciences IP Limited except certain content provided by third parties. Reaxys is a trademark of Elsevier Life Sciences IP Limited.

3/10

2018-07-09 14:42:02


Quantitative value

100

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 3 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Minimum inhibitory concentration of the compound dissolved in DMSO against Staphylococcus aureus ATCC 29213 by disk diffusion susceptibility assay

Biological Species/NCBI ID

Staphylococcus aureus ATCC 29213

Substance RN

3145953View in Reaxys

Measurement Parameter

MIC

Unit

µg

Measurement Object

Minimum Inhibitory Concentration

Qualitative value

>

Quantitative value

100

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 4 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Minimum inhibitory concentration of the compound dissolved in DMSO against Cryptococcus neoformans ATCC 90112 by disk diffusion susceptibility assay

Biological Species/NCBI ID

Cryptococcus neoformans ATCC 90112

Substance RN

3145953View in Reaxys

Measurement Parameter

MIC

Unit

µg

Measurement Object

Minimum Inhibitory Concentration

Qualitative value

>

Quantitative value

100

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 5 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Growth inhibition of the compound against human ovary cancer OVCAR-3 cells

Biological Species/NCBI ID

human

Cells/Cell Lines

OVCAR-3 cell line

Substance RN

3145953View in Reaxys

Measurement Parameter

GI50

Unit

µg/mL

Measurement Object

Growth inhibition

Qualitative value

=

Quantitative value

0.42

Measurement pX

5.75

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 6 of 21

Bioassay Category

In Vitro (Efficacy)

Copyright © 2018 Elsevier Life Sciences IP Limited except certain content provided by third parties. Reaxys is a trademark of Elsevier Life Sciences IP Limited.

4/10

2018-07-09 14:42:02


Bioassay Details

Minimum inhibitory concentration of the compound dissolved in DMSO against Enterococcus faecalis ATCC 29212 by disk diffusion susceptibility assay

Biological Species/NCBI ID

Enterococcus faecalis ATCC 29212

Substance RN

3145953View in Reaxys

Measurement Parameter

MIC

Unit

µg

Measurement Object

Minimum Inhibitory Concentration

Qualitative value

>

Quantitative value

100

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 7 of 21

Substance Action on Target

Inhibitor

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Growth inhibition of the compound against human prostate cancer DU-145 cells

Biological Species/NCBI ID

human

Cells/Cell Lines

DU145 cell line

Substance RN

3145953View in Reaxys

Qualitative Results

NA = Not available

Measurement Parameter

GI50

Measurement Object

Growth inhibition

Qualitative value

ND

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 8 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Minimum inhibitory concentration of the compound dissolved in DMSO against Enterobacter cloacae ATCC 13047 by disk diffusion susceptibility assay

Biological Species/NCBI ID

Enterobacter cloacae ATCC 13047

Substance RN

3145953View in Reaxys

Measurement Parameter

MIC

Unit

µg

Measurement Object

Minimum Inhibitory Concentration

Qualitative value

>

Quantitative value

100

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 9 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Growth inhibition of the compound against human breast cancer MCF-7 cells; NA = Not available

Biological Species/NCBI ID

human

Cells/Cell Lines

MCF-7 cell line

Substance RN

3145953View in Reaxys

Copyright © 2018 Elsevier Life Sciences IP Limited except certain content provided by third parties. Reaxys is a trademark of Elsevier Life Sciences IP Limited.

5/10

2018-07-09 14:42:02


Qualitative Results

NA = Not available

Measurement Parameter

GI50

Measurement Object

Growth inhibition

Qualitative value

ND

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 10 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Minimum inhibitory concentration of the compound dissolved in DMSO against Streptococcus pneumoniae ATCC 6303 by disk diffusion susceptibility assay

Biological Species/NCBI ID

Streptococcus pneumoniae ATCC 6303

Substance RN

3145953View in Reaxys

Measurement Parameter

MIC

Unit

µg

Measurement Object

Minimum Inhibitory Concentration

Qualitative value

>

Quantitative value

100

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 11 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Growth inhibition of the compound against human melanoma cancer SK-MEL-5 cells

Biological Species/NCBI ID

human

Cells/Cell Lines

SK-MEL-5 cell line

Substance RN

3145953View in Reaxys

Measurement Parameter

GI50

Unit

µg/mL

Measurement Object

Growth inhibition

Qualitative value

=

Quantitative value

0.61

Measurement pX

5.59

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 12 of 21

Substance Action on Target

Inhibitor

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Growth inhibition of the compound against human pancreatic cancer BXPC-3 cells; NA = Not available

Biological Species/NCBI ID

human

Cells/Cell Lines

BxPC-3 cell line

Substance RN

3145953View in Reaxys

Qualitative Results

NA = Not available

Measurement Parameter

GI50

Copyright © 2018 Elsevier Life Sciences IP Limited except certain content provided by third parties. Reaxys is a trademark of Elsevier Life Sciences IP Limited.

6/10

2018-07-09 14:42:02


Measurement Object

Growth inhibition

Qualitative value

ND

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 13 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Effective dose of the compound against murine leukemia P388 cells

Biological Species/NCBI ID

mouse

Cells/Cell Lines

P388 cell line

Substance RN

3145953View in Reaxys

Measurement Parameter

EC50

Unit

µg/mL

Measurement Object

Effective dose

Qualitative value

=

Quantitative value

14

Measurement pX

4.23

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 14 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Growth inhibition of the compound against human CNS cancer SF268 cells; NA = Not available

Biological Species/NCBI ID

human

Cells/Cell Lines

SF268 cell line

Substance RN

3145953View in Reaxys

Qualitative Results

NA = Not available

Measurement Parameter

GI50

Measurement Object

Growth inhibition

Qualitative value

ND

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 15 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Minimum inhibitory concentration of the compound dissolved in DMSO against Neisseria gonorrhoeae ATCC 49226 by disk diffusion susceptibility assay

Biological Species/NCBI ID

Neisseria gonorrhoeae ATCC 49226

Substance RN

3145953View in Reaxys

Measurement Parameter

MIC

Unit

µg

Measurement Object

Minimum Inhibitory Concentration

Qualitative value

>

Quantitative value

100

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys

Copyright © 2018 Elsevier Life Sciences IP Limited except certain content provided by third parties. Reaxys is a trademark of Elsevier Life Sciences IP Limited.

7/10

2018-07-09 14:42:02


16 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Growth inhibition of the compound against human colon cancer KM20L2 cells

Biological Species/NCBI ID

human

Cells/Cell Lines

KM20L2 cell line

Substance RN

3145953View in Reaxys

Measurement Parameter

GI50

Unit

µg/mL

Measurement Object

Growth inhibition

Qualitative value

=

Quantitative value

0.38

Measurement pX

5.8

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 17 of 21

Substance Action on Target

Inhibitor

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Growth inhibition of the compound against human renal cancer A498 cells

Biological Species/NCBI ID

human

Cells/Cell Lines

A-498 cell line

Substance RN

3145953View in Reaxys

Measurement Parameter

GI50

Unit

µg/mL

Measurement Object

Growth inhibition

Qualitative value

=

Quantitative value

0.36

Measurement pX

5.82

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 18 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Growth inhibition of the compound against human lung-NSC cancer NCI-H460 cells

Biological Species/NCBI ID

human

Cells/Cell Lines

NCI-H460 cell line

Substance RN

3145953View in Reaxys

Measurement Parameter

GI50

Unit

µg/mL

Measurement Object

Growth inhibition

Qualitative value

=

Quantitative value

0.32

Measurement pX

5.87

Copyright © 2018 Elsevier Life Sciences IP Limited except certain content provided by third parties. Reaxys is a trademark of Elsevier Life Sciences IP Limited.

8/10

2018-07-09 14:42:02


Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 19 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Growth inhibition of the compound against human CNS cancer SF295 cells

Biological Species/NCBI ID

human

Cells/Cell Lines

SF295 cell line

Substance RN

3145953View in Reaxys

Measurement Parameter

GI50

Unit

µg/mL

Measurement Object

Growth inhibition

Qualitative value

=

Quantitative value

0.45

Measurement pX

5.73

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 20 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Minimum inhibitory concentration of the compound dissolved in DMSO against Candida albicans ATCC 90028 by disk diffusion susceptibility assay

Biological Species/NCBI ID

Candida albicans ATCC 90028

Substance RN

3145953View in Reaxys

Measurement Parameter

MIC

Unit

µg

Measurement Object

Minimum Inhibitory Concentration

Qualitative value

>

Quantitative value

100

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys 21 of 21

Bioassay Category

In Vitro (Efficacy)

Bioassay Details

Minimum inhibitory concentration of the compound dissolved in DMSO against Micrococcus luteus presque isle 456 by disk diffusion susceptibility assay

Biological Species/NCBI ID

Micrococcus luteus Presque Isle 456

Substance RN

3145953View in Reaxys

Measurement Parameter

MIC

Unit

µg

Measurement Object

Minimum Inhibitory Concentration

Qualitative value

>

Quantitative value

100

Pettit, Robin K.; Pettit, George R.; Hamel, Ernest; Hogan, Fiona; Moser, Bryan R.; Wolf, Sonja; Pon, Sandy; Chapuis, Jean-Charles; Schmidt, Jean M.; Bioorganic and Medicinal Chemistry; vol. 17; nb. 18; (2009); p. 6606 - 6612, View in Reaxys

Copyright © 2018 Elsevier Life Sciences IP Limited except certain content provided by third parties. Reaxys is a trademark of Elsevier Life Sciences IP Limited.

9/10

2018-07-09 14:42:02


Reaxys ID 8546971 View in Reaxys O

2/2 Chemical Name: 1,3,5-trimethoxy-2-(2-nitrovinyl)benzene Linear Structure Formula: C11H13NO5 Molecular Formula: C11H13NO5 Molecular Weight: 239.228 Type of Substance: isocyclic InChI Key: URHPFHDNYKOMAI-UHFFFAOYSA-N Note:

O N

O

O

O

Substance Label (4) Label References 1

Jiang, Chen-Ran; Zhao, Chun-Liang; Guo, Hui-Fang; He, Wei; Chemical Communications; vol. 52; nb. 50; (2016); p. 7862 - 7865, View in Reaxys

9c

Kazin, Nikita A.; Kvashnin, Yuriy A.; Irgashev, Roman A.; Dehaen, Wim; Rusinov, Gennady L.; Charushin, Valery N.; Tetrahedron Letters; vol. 56; nb. 14; (2015); p. 1865 - 1869, View in Reaxys

9

Patent; PIRAMAL LIFE SCIENCES LIMITED; BANDGAR, Babasaheb Pandurang; TOTRE, Jalindar Vasant; WO2011/121505; (2011); (A1) English, View in Reaxys

t.,pr.,sr.no.3

Bandgar; Uppalla; Synthetic Communications; vol. 30; nb. 12; (2000); p. 2071 - 2075, View in Reaxys

Druglikeness (1) 1 of 1

LogP

2.242

H Bond Donors

0

H Bond Acceptors

0

Rotatable Bonds

5

TPSA

73.51

Lipinski Number

4

Veber Number

2

NMR Spectroscopy (1) 1 of 1

Nucleus (NMR Spectroscopy)

1H

Solvents (NMR Spectroscopy)

chloroform-d1

Original Text (NMR Spectroscopy)

1

Location

Page/Page column 42

Comment (NMR Spectroscopy)

Signals given

HNMR (CDCI3): β 8.53 (d, 1 H), 8.0 (d, 1 H), 6.1 1 (s, 2H), 3.90 (s, 6H), 3.87 (s, 3H);

Patent; PIRAMAL LIFE SCIENCES LIMITED; BANDGAR, Babasaheb Pandurang; TOTRE, Jalindar Vasant; WO2011/121505; (2011); (A1) English, View in Reaxys Mass Spectrometry (1) Location References Page/Page column 42

Patent; PIRAMAL LIFE SCIENCES LIMITED; BANDGAR, Babasaheb Pandurang; TOTRE, Jalindar Vasant; WO2011/121505; (2011); (A1) English, View in Reaxys

Copyright © 2018 Elsevier Life Sciences IP Limited except certain content provided by third parties. Reaxys is a trademark of Elsevier Life Sciences IP Limited.

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