Basics of Duchenne

Page 1


Duchenne muscular dystrophy

? Annemieke Aartsma-Rus


Overview Â

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Genes and proteins

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Muscles Â

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Muscles Â

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Muscle fibers

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Dystrophin Â

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Genes and proteins

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Gene  Protein Cell nucleus DNA Temporary gene copy (RNA) Cell body (cytoplasm)

Protein factory

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Dystrophin  gene Â

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Splicing  2

1

6

3 5

7

4

1

2

3

4

5

6

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7

1 2 3 4 5 6 7 8 1 - - - - - - - - - 79


Duchenne: geneHc code disrupted

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Duchenne: geneHc code disrupted Exon 46

Exon 47

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?

Exon 51

Exon 52


Consequence Â

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Becker: geneHc code maintained

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Becker: geneHc code maintained Exon 46

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Exon 47

Exon 52

Exon 53


Duchenne: no funcHonal dystrophin

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No funcHonal dystrophin No dystrophin

Leaky muscle fibers

Calcium leaks into fibers AcHvaHon proteases

Damage energy producing organels

More muscle damage

InflammaHon Scar Hssue

Less muscle regeneraHon

Loss of muscle fibers Loss of muscle func/on Annemieke Aartsma-Rus


Therapy No dystrophin

Leaky muscle fibers

Calcium leaks into fibers AcHvaHon proteases

Damage energy producing organels

More muscle damage

InflammaHon Scar Hssue

Less muscle regeneraHon

Loss of muscle fibers Loss of muscle func/on Annemieke Aartsma-Rus


CorHcosteroids No dystrophin

Leaky muscle fibers

Calcium leaks into fibers AcHvaHon proteases

Damage energy producing organels

More muscle damage

InflammaHon Scar Hssue

Less muscle regeneraHon

Loss of muscle fibers reduced Loss of muscle func/on reduced Annemieke Aartsma-Rus


Reduce muscle fiber damage No dystrophin

Leaky muscle fibers

Calcium leaks into fibers AcHvaHon proteases

Damage energy producing organels

More muscle damage

InflammaHon Scar Hssue

Less muscle regeneraHon

Loss of muscle fibers reduced Loss of muscle func/on reduced Annemieke Aartsma-Rus


Increase muscle mass No dystrophin

Leaky muscle fibers

Loss of muscle fibers compensated Loss of muscle funcHon compensated Annemieke Aartsma-Rus


Utrophin upregulaHon

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Utrophin upregulaHon No dystrophin

Leaky muscle fibers

Loss of muscle fibers prevented Loss of muscle func/on prevented Annemieke Aartsma-Rus


Gene therapy No dystrophin

Leaky muscle fibers

Loss of muscle fibers prevented Loss of muscle func/on prevented Annemieke Aartsma-Rus


Cell therapy No dystrophin

Leaky muscle fibers

Loss of muscle fibers prevented Loss of muscle func/on prevented Annemieke Aartsma-Rus


Terms/jargon: cell models

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Terms/jargon: animal models

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Terms/jargon: animal models

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Terms/jargon Â

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Terms/jargon Â

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Terms/jargon Dystrophin immune staining Healthy

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Mdx mouse

Duchenne


Terms/jargon Â

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Terms/jargon Â

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Terms/jargon Â

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Summary/Outlook Â

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More  informaHon Â

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Thank you!

Annemieke Aartsma-Rus


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