PHARM CHAPTER 11 2008

Page 1

DRUGS FOR SEIZURES

Chapter 11


INTRODUCTION  Epilepsy

is a common disorder of the CNS characterized by symptoms of blackout, fainting spells, apparent clumsiness, temporary loss of memory, and/or irregular seizure activity.


INTRODUCTION  Over

two million Americans have epilepsy, and except for when these symptoms are expressed, most of the time it appears that their health is not challenged.


SEIZURES & CONVULSIONS ARE SYMPTOMS OF EPILEPSY Seizures—abnormal or uncontrollable neuronal discharges within the brain.  May cause a blank stare, a loss of consciousness, jerking body movements, or a period of general confusion for the client. 


SEIZURES & CONVULSIONS  The

terms convulsion and seizure are not the same.  Convulsions specifically refer to involuntary, violent spasms of the large skeletal muscles of the face, neck, arms, and legs.


SEIZURES & CONVULSIONS All convulsions are seizures, but not all seizures are convulsions.  Although some types of seizures do indeed involve convulsions, other seizures do not.  Thus antiseizure meds rather than anticonvulsants. 


CAUSES       

Neuronal damage or injury Head trauma Extreme fever Heat exhaustion Brain tumor Infections Stroke

Lowered blood glucose  High protein levels  Mood disorder, antipsychotic, and local anesthetic med’s  Drug abuse—cocaine  Alcohol withdrawal  Withdrawal from sedative-hypnotics 


TYPES OF SEIZURES  Partial  

seizures

Simple Complex

 Generalized    

seizures

Absence (petit mal) Atonic seizure (drop attacks) Myoclonic seizure Tonic-clonic (grand mal)


STATUS EPILEPTICUS  Status

epilepticus is a medical emergency brought on by repeated generalized seizures and convulsions.  Muscle spasms may block the airway, depriving the brain of oxygen.


SEIZURE MANAGEMENT Effective seizure management involves strict adherence to drug therapy.  Choice of drug depends on the type of seizures, medical history, diagnostic studies, and the pathological processes causing the seizures. 


SEIZURE MANAGEMENT 

Because seizures are likely to occur with abrupt withdrawal, antiseizure medications is withdrawn over a period of 6 to 12 weeks.

In most cases, a single drug effectively manages seizures.  Once seizures are controlled, patients are continued indefinitely on the antiseizure drug 


SEIZURE MANAGEMENT  Withdrawal

should only be attempted after at least 3 years of being seizure free, and only under the close observation and direction of the healthcare team.


SEIZURE MANAGEMENT  Goal

of antiseizure drug therapy is to suppress neuronal activity just enough to prevent abnormal or repetitive firing.


DRUGS WITH GABA ACTION  Drugs

with GABA action are drugs with the ability to mimic effects of the inhibitory neurotransmitter GABA.  Ex. Benzodiazepines, barbiturates, and miscellaneous drugs  DP-phenobarbital (luminal) pg. 182.


PHENYTOIN AND PHEYTOIN-LIKE DRUGS (HYDANTOINS) Delay influx of sodium ions across neuronal membrane.  Ex.—hydantoins, carbamazepine (Tegretol), divalproex (Depakote), valoproic acid (Depakene)  DP for phenytoin—Dilantin pg. 185  DP for valoproic acid (Depakene) pg. 185 


SUCCINIMIDES  Succinimides

delay entry of calcium ions into neuron— increases electrical threshold; no impulse transmitted  DP—ethosuximide (Zarontin) pg. 186.


SOME CONTROLLED BY A PREFERRED GROUP OF DRUGS  Drugs

do not cure epilepsy; just reduce number of seizures.  Same seizures do not respond to same drug.


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